SCHEMBL8208288

SCHEMBL8208288

CNC(=O)CN1C(=O)C2(CCN(C(=O)OC(C)(C)C)CC2)C1c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
KDM4E B2RXH2 1/20 0.43
PKM P14618 1/20 0.43
TRPV1 Q8NER1 3/20 0.42
TSHR P16473 2/20 0.42
ALOX15 P16050 1/20 0.42
ATM Q13315 1/20 0.42
GPR119 Q8TDV5 2/20 0.42
TACR1 P25103 1/20 0.41
KDM1A O60341 2/20 0.41
STS P08842 1/20 0.41
USP30 Q70CQ3 1/20 0.41
NR1H2 P55055 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8224879 0.86 HDAC1 (0.44) HDAC1HDAC6KDM4EPKMTRPV1
SCHEMBL8218924 0.83 HDAC1 (0.47) HDAC1HDAC6KDM4EPKMTRPV1
SCHEMBL8227850 0.81 HDAC1 (0.45) HDAC1HDAC6KDM4EPKMTRPV1
SCHEMBL8218899 0.80 GPR119 (0.48) HDAC1HDAC6KDM4EPKMTRPV1
SCHEMBL8218912 0.80 HDAC1 (0.46) HDAC1HDAC6KDM4EPKMTRPV1
SCHEMBL8212694 0.78 TRPV1 (0.61) HDAC1HDAC6TRPV1TSHRALOX15
SCHEMBL8200179 0.78 TSHR (0.47) KDM4EPKMTRPV1TSHRALOX15
SCHEMBL8224883 0.77 GPR119 (0.43) HDAC1HDAC6GPR119
SCHEMBL14263479 0.76 MEN1 (0.43) HDAC1HDAC6STS
SCHEMBL8227881 0.75 HDAC1 (0.55) HDAC1HDAC6KDM4EGPR119KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033465-A1 AZETIDINONE DERIVATIVES AND METHODS OF USE THEREOF SCHERING CORPORATION (US) 2008-03-20 WO disclosed