Trifluoroacetamide

Trifluoroacetamide

SCHEMBL8213276

CC[C@H](NC(=O)OC(C)(C)C)C(=O)N1c2ccc(Cl)cc2C[C@H]1C(=O)O.NC(=O)C(F)(F)F

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.40
MC4R P32245 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
ALOX12 P18054 1/20 0.37
CTSL P07711 1/20 0.36
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
ACE P12821 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5563362 0.94 MC4R (0.42) SCN9AMC4RKDM4EALDH1A1GAA
SCHEMBL7668349 0.94 MC4R (0.42) SCN9AMC4RKDM4EALDH1A1GAA
2,2,2-Trifluoroethanaminium SCHEMBL8213280 0.93 SCN9A (0.40) SCN9AMC4RKDM4EALDH1A1GAA
Trifluoroacetamide SCHEMBL8207815 0.88 SCN9A (0.35) SCN9AACE
SCHEMBL5563656 0.87 MC4R (0.41) SCN9AMC4RKDM4EALDH1A1GAA
SCHEMBL5563441 0.86 MC4R (0.41) SCN9AMC4RKDM4EALDH1A1GAA
SCHEMBL5568361 0.85 ACE (0.40) ACE
SCHEMBL5568442 0.83 SCN9A (0.37) SCN9AACE
SCHEMBL5563792 0.83 SCN9A (0.37) SCN9AACE
Trifluoroacetamide SCHEMBL8210338 0.83 ACE (0.39) SCN9AMC4RACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042288-A1 TRIPEPTIDYL PEPTIDASE INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2000-10-11 EP disclosed
WO-1999033801-A1 TRIPEPTIDYL PEPTIDASE INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1999-07-08 WO disclosed