SCHEMBL8213620

SCHEMBL8213620

CC(F)(F)COC(=O)N1C[C@H](N)C(=O)N(CC(F)(F)F)c2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 12/20 0.37
SCN10A Q9Y5Y9 1/20 0.35
XIAP P98170 1/20 0.32
KCNH2 Q12809 2/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
KDM1A O60341 1/20 0.31
AADAT Q8N5Z0 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4565038 0.92 SCN9A (0.35) SCN9ASCN10AXIAPKCNH2AADAT
Hydrochloric Acid SCHEMBL4565037 0.91 SCN9A (0.34) SCN9ASCN10AXIAPKCNH2AADAT
Hydrochloric Acid SCHEMBL4992340 0.91 SCN9A (0.34) SCN9ASCN10AXIAPKCNH2AADAT
SCHEMBL4434484 0.85 SCN9A (0.38) SCN9ASCN10AKCNH2
Hydrochloric Acid SCHEMBL4434476 0.84 SCN9A (0.38) SCN9ASCN10AKCNH2
Hydrochloric Acid SCHEMBL4434487 0.84 SCN9A (0.38) SCN9ASCN10AKCNH2
SCHEMBL4434152 0.83 NOTUM (0.42) SCN9ASCN10AXIAPKCNH2
Hydrochloric Acid SCHEMBL4429066 0.82 NOTUM (0.41) SCN9ASCN10AXIAPKCNH2
Hydrochloric Acid SCHEMBL4429072 0.82 NOTUM (0.41) SCN9ASCN10AXIAPKCNH2
SCHEMBL4992925 0.78 NR1H2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008034735-A2 4-OXO-2,3,4,5-TETRAHYDRO-BENZO[B][1,4]DIAZEPINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO disclosed