SCHEMBL4434152

SCHEMBL4434152

CC(=O)N1C[C@H](N)C(=O)N(CC(F)(F)F)c2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 5/20 0.42
BRD4 O60885 2/20 0.41
XIAP P98170 3/20 0.38
POLB P06746 1/20 0.37
SCN9A Q15858 5/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KCNH2 Q12809 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4429066 0.99 NOTUM (0.41) NOTUMBRD4XIAPPOLBSCN9A
Hydrochloric Acid SCHEMBL4429072 0.99 NOTUM (0.41) NOTUMBRD4XIAPPOLBSCN9A
Hydrochloric Acid SCHEMBL5541728 0.84 MAT2A (0.39) BRD4POLBSCN9AALDH1A1KCNH2
SCHEMBL4425590 0.84 NOTUM (0.46) NOTUMBRD4XIAPPOLBALDH1A1
SCHEMBL4425596 0.84 NOTUM (0.46) NOTUMBRD4XIAPPOLBALDH1A1
SCHEMBL4565038 0.83 SCN9A (0.35) XIAPSCN9AKCNH2SCN10A
SCHEMBL8213620 0.83 SCN9A (0.37) XIAPSCN9AKCNH2SCN10A
SCHEMBL14599943 0.83 XIAP (0.43) NOTUMBRD4XIAPPOLBSCN9A
Hydrochloric Acid SCHEMBL4565037 0.82 SCN9A (0.34) XIAPSCN9AKCNH2SCN10A
Hydrochloric Acid SCHEMBL4992340 0.82 SCN9A (0.34) XIAPSCN9AKCNH2SCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711470-B1 MALONAMIDE DERIVATIVES BLOCKING THE ACTIVTIY OF GAMMA-SECRETASE HOFFMANN LA ROCHE (CH) 2009-04-15 EP disclosed