SCHEMBL8214899

SCHEMBL8214899

CCn1c(N2CCC[C@@H](N)C2)cc2c1c(=O)n(Cc1ccc3ncccc3n1)c(=O)n2C

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.51
CYP3A4 P08684 10/20 0.51
KCNH2 Q12809 2/20 0.48
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
DPP9 Q86TI2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12047556 0.91 DPP4 (0.62) DPP4CYP3A4KCNH2DPP9
SCHEMBL8216727 0.86 DPP4 (0.49) DPP4CYP3A4CYP1A2CYP2D6
SCHEMBL11910982 0.86 DPP4 (0.65) DPP4DPP9
SCHEMBL8215317 0.83 DPP4 (0.48) DPP4CYP3A4KCNH2CYP1A2CYP2D6
SCHEMBL8206433 0.82 DPP4 (0.63) DPP4CYP3A4KCNH2CYP1A2CYP2D6
SCHEMBL8206963 0.82 DPP4 (0.62) DPP4CYP3A4KCNH2CYP1A2CYP2D6
SCHEMBL8213697 0.82 DPP4 (0.69) DPP4KCNH2
SCHEMBL12060339 0.82 DPP4 (0.49) DPP4CYP3A4KCNH2DPP9
SCHEMBL8216730 0.81 DPP4 (0.63) DPP4CYP3A4KCNH2DPP9
SCHEMBL8215864 0.81 DPP4 (0.52) DPP4CYP3A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008017670-A1 PYRROLO [3, 2 -D] PYRIMIDINES AS DPP-IV INHIBITORS FOR THE TREATMENT OF DIABETES MELLITUS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-02-14 WO disclosed