SCHEMBL8216007

SCHEMBL8216007

CCCC1CC(NC(=O)c2cccc3oc(N4CCOC[C@@H]4CCC)nc23)CC(C)N1C

nearest known ligand 0.80

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 20/20 0.80
KCNH2 Q12809 3/20 0.57
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8214885 0.96 HTR3A (0.74) HTR3AKCNH2CYP2C19
SCHEMBL3986685 0.89 HTR3A (1.00) HTR3AKCNH2CYP2C19
SCHEMBL1004948 0.89 HTR3A (1.00) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1007726 0.88 HTR3A (0.98) HTR3AKCNH2CYP2C19
SCHEMBL8224160 0.84 HTR3A (0.71) HTR3AKCNH2CYP2C19
SCHEMBL8215391 0.82 HTR3A (0.55) HTR3AKCNH2CYP2C19
SCHEMBL1005577 0.82 HTR3A (1.00) HTR3AKCNH2CYP2C19
SCHEMBL1006203 0.82 HTR3A (1.00) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1005983 0.81 HTR3A (0.98) HTR3AKCNH2CYP2C19
SCHEMBL1007048 0.81 HTR3A (0.67) HTR3AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed