SCHEMBL8216643

SCHEMBL8216643

COc1cc(-n2cccn2)ccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.53
RXRA P19793 4/20 0.50
GRIN1 Q05586 4/20 0.50
GRIN2B Q13224 4/20 0.50
MET P08581 1/20 0.43
MAPT P10636 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPK1 P28482 1/20 0.41
PTPN1 P18031 1/20 0.41
HCRTR1 O43613 4/20 0.41
HCRTR2 O43614 4/20 0.41
CCNT1 O60563 1/20 0.41
CDK9 P50750 1/20 0.41
DYRK1A Q13627 1/20 0.40
EGLN2 Q96KS0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195797 0.88 NOTUM (0.53) NOTUMMAPTKDM4EALDH1A1MAPK1
SCHEMBL27932708 0.85 NOTUM (0.49) NOTUMMAPTKDM4EALDH1A1MAPK1
SCHEMBL13347571 0.83 NOTUM (0.46) NOTUMMAPTKDM4EALDH1A1MAPK1
SCHEMBL2188351 0.81 NLRP3 (0.45) NOTUMKDM4EALDH1A1MAPK1PTPN1
SCHEMBL5756029 0.81 PTPN1 (0.49) NOTUMMAPTKDM4EALDH1A1MAPK1
SCHEMBL15475872 0.81 PTPN1 (0.49) NOTUMKDM4EALDH1A1MAPK1PTPN1
SCHEMBL8114245 0.81 NOTUM (0.45) NOTUMMAPTKDM4EALDH1A1MAPK1
SCHEMBL28677811 0.81 GRIN1 (0.53) NOTUMRXRAGRIN1GRIN2B
SCHEMBL13310513 0.81 NOTUM (0.45) NOTUMMAPTKDM4EALDH1A1MAPK1
SCHEMBL11337325 0.80 NOTUM (0.63) NOTUMMAPTKDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed