SCHEMBL8220977

SCHEMBL8220977

N#Cc1ccc(C2N(c3ccc(F)c(Cl)c3)C(=O)C23CCNCC3)cc1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 10/20 0.47
MDM2 Q00987 8/20 0.39
ITGB2 P05107 1/20 0.39
ICAM1 P05362 1/20 0.39
ITGAL P20701 1/20 0.39
TP53 P04637 4/20 0.38
IDO1 P14902 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12844640 0.88 CACNA1H (0.49) CACNA1HMDM2TP53
SCHEMBL12844637 0.88 CACNA1H (0.43) CACNA1HITGB2ICAM1ITGAL
SCHEMBL8210807 0.85 CACNA1H (0.47) CACNA1HMDM2TP53
SCHEMBL8209942 0.78 HSD11B1 (0.50) CACNA1H
SCHEMBL8229542 0.77 CACNA1H (0.71) CACNA1HMDM2
SCHEMBL3998065 0.76 CACNA1H (0.66) CACNA1H
SCHEMBL8201959 0.76 CACNA1H (0.62) CACNA1H
SCHEMBL12890364 0.73 CACNA1H (0.40) CACNA1H
SCHEMBL8212780 0.73 CACNA1H (0.53) CACNA1HMDM2TP53
SCHEMBL12777757 0.71 HSD11B1 (0.50) CACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033468-A2 AZETIDINE AND AZETIDONE DERIVATIVES USEFUL IN TREATING PAIN AND DISORDERS OF LIPID METABOLISM SCHERING CORPORATION (US) 2008-03-20 WO disclosed