Bicuculline

Bicuculline

SCHEMBL8222

CN1CCc2cc3c(cc2[C@H]1[C@@H]1OC(=O)c2c1ccc1c2OCO1)OCO3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 1.00
CYP2C9 P11712 6/20 1.00
CYP2C19 P33261 6/20 1.00
CYP2D6 P10635 6/20 1.00
TSHR P16473 4/20 1.00
CYP1A2 P05177 3/20 1.00
LMNA P02545 3/20 1.00
HIF1A Q16665 1/20 1.00
GABRP O00591 1/20 1.00
GABRD O14764 1/20 1.00
GABRA1 P14867 1/20 1.00
GABRB1 P18505 1/20 1.00
GABRG2 P18507 1/20 1.00
GABRB3 P28472 1/20 1.00
GABRA5 P31644 1/20 1.00
GABRA3 P34903 1/20 1.00
GABRA2 P47869 1/20 1.00
GABRB2 P47870 1/20 1.00
GABRA4 P48169 1/20 1.00
GABRE P78334 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicuculline SCHEMBL28213750 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL29652597 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL29617593 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL29390611 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL7913545 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL5481014 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL5783586 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL29366341 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL16320040 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL2532354 0.99 CYP3A4 (0.98) CYP3A4CYP2C9CYP2C19CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3357 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4717276-A2 OPHTHALMIC COMPOSITIONS COMPRISING LEVODOPA, AN ANTIOXIDANT AND AN AQUEOUS CARRIER University of Canberra (AU) 2026-04-01 EP claimed
EP-3442516-B1 OPHTHALMIC COMPOSITIONS COMPRISING LEVODOPA, AN ANTIOXIDANT AND AN AQUEOUS CARRIER UNIV CANBERRA (AU) 2025-11-12 EP claimed
CN-119409583-A Beta-chiral tertiary amine compound and preparation method thereof 同济大学 2025-02-11 CN claimed
WO-2025024501-A1 NEUROMODULATORY PEPTIDES LACTOCORE, INC. (US) 2025-01-30 WO claimed
US-12194201-B2 Silica nanoparticle doped conductive polymer University of Pittsburgh—of the Commonwealth System of Higher Education (US) 2025-01-14 US claimed
US-20240390364-A1 Novel Pyridine Compositions and their use in methods for preventing or treating diseases, disorders and conditions REID CHRISTOPHER BRIAN (US) 2024-11-28 US claimed
CN-112770734-B Inhibition method 堪培拉大学 2024-08-20 CN claimed
CN-118286599-A Method for regulating and controlling epileptiform discharge and researching mechanism by micron-scale electrical stimulation 天津工业大学 2024-07-05 CN claimed
CN-118105389-A Composition for nerve block surgery and application of composition in preparation of medicines 中国人民解放军战略支援部队特色医学中心 2024-05-31 CN claimed
US-11890266-B2 Ophthalmic compositions including levodopa, an antioxidant and an aqueous carrier UNIVERSITY OF CANBERRA (AU) 2024-02-06 US claimed
US-20040177398-A1 Regulation of plant fertility by modulation of GABA levels in flowers CHICAGO, THE UNIVERSITY OF 2004-09-09 US claimed
WO-2004068137-A2 METHODS AND DEVICE FOR IN VITRO DETECTION AND CHARACTERIZATION OF PSYCHOACTIVES USING ANALYSIS OF REPETITIVE ELECTRICAL ACTIVITY IN A NEURONAL SAMPLE MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2004-08-12 WO claimed
US-20040137515-A1 Methods and device for in vitro detection and characterization of psychoactives using analysis of repetitive electrical activity in a neuronal sample MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. (JP) 2004-07-15 US claimed
EP-1416794-A2 REGULATION OF PLANT FERTILITY BY MODULATION OF GABA LEVELS IN FLOWERS The University of Chicago (US) 2004-05-12 EP claimed
EP-1303280-A1 ENHANCED BRAIN FUNCTION BY GABA-ERGIC STIMULATION University of Utah Research Foundation (US) 2003-04-23 EP claimed
WO-2003000039-A2 REGULATION OF PLANT FERTILITY BY MODULATION OF GABA LEVELS IN FLOWERS UNIVERSITY OF CHICAGO (US) 2003-01-03 WO claimed
US-20020156016-A1 Control of cell growth by altering cell membrane potentials MANITOBA, UNIVERSITY OF, THE (CA) 2002-10-24 US claimed
WO-2002000221-A1 ENHANCED BRAIN FUNCTION BY GABA-ERGIC STIMULATION UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2002-01-03 WO claimed
WO-2001008670-A2 METHODS AND COMPOSITIONS FOR ALLEVIATING STUTTERING INTERNEURON PHARMACEUTICALS, INC. (US) 2001-02-08 WO claimed
CN-1091637-A Application of dicentrine in treating benign prostatic hyperplasia DENG ZHEMING (CN) 1994-09-07 CN claimed