Bicuculline

Bicuculline

SCHEMBL7913545

CN1CCc2cc3c(cc2[C@H]1[C@H]1OC(=O)c2c1ccc1c2OCO1)OCO3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 1.00
CYP2C9 P11712 6/20 1.00
CYP2C19 P33261 6/20 1.00
CYP2D6 P10635 6/20 1.00
TSHR P16473 4/20 1.00
CYP1A2 P05177 3/20 1.00
LMNA P02545 3/20 1.00
HIF1A Q16665 1/20 1.00
GABRP O00591 1/20 1.00
GABRD O14764 1/20 1.00
GABRA1 P14867 1/20 1.00
GABRB1 P18505 1/20 1.00
GABRG2 P18507 1/20 1.00
GABRB3 P28472 1/20 1.00
GABRA5 P31644 1/20 1.00
GABRA3 P34903 1/20 1.00
GABRA2 P47869 1/20 1.00
GABRB2 P47870 1/20 1.00
GABRA4 P48169 1/20 1.00
GABRE P78334 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicuculline SCHEMBL28213750 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL29652597 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL29617593 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL29390611 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL5481014 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL5783586 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL8222 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL29366341 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL16320040 1.00 CYP3A4 (1.00) CYP3A4CYP2C9CYP2C19CYP2D6TSHR
Bicuculline SCHEMBL2532354 0.99 CYP3A4 (0.98) CYP3A4CYP2C9CYP2C19CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 78 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023219526-A1 MULTITARGET ANTIVIRAL DIETARY SUPPLEMENT PROKIN MILAN (RS) 2023-11-16 WO claimed
US-20260103736-A1 Methods Of Improving Production Of Morphinan Alkaloids And Derivatives ANTHEIA INC (US) 2026-04-16 US disclosed
US-12497638-B2 Methods of producing epimerases and benzylisoquinoline alkaloids THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2025-12-16 US disclosed
EP-4594342-A2 METHODS OF IMPROVING PRODUCTION OF MORPHINAN ALKALOIDS AND DERIVATIVES Antheia, Inc. (US) 2025-08-06 EP disclosed
EP-3221461-B1 NOSCAPINOID-PRODUCING MICROBES AND METHODS OF MAKING AND USING THE SAME UNIV LELAND STANFORD JUNIOR (US) 2025-01-01 EP disclosed
US-20240218408-A1 Methods of Producing Epimerases and Benzylisoquinoline Alkaloids HERCULES CAPITAL, INC., AS AGENT 2024-07-04 US disclosed
WO-2024073755-A2 METHODS OF IMPROVING PRODUCTION OF MORPHINAN ALKALOIDS AND DERIVATIVES ANTHEIA, INC. (US) 2024-04-04 WO disclosed
US-20240102061-A1 METHODS OF IMPROVING PRODUCTION OF MORPHINAN ALKALOIDS AND DERIVATIVES HERCULES CAPITAL, INC., AS AGENT 2024-03-28 US disclosed
US-11859225-B2 Methods of producing epimerases and benzylisoquinoline alkaloids THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2024-01-02 US disclosed
WO-2023219526-A1 MULTITARGET ANTIVIRAL DIETARY SUPPLEMENT PROKIN MILAN (RS) 2023-11-16 WO disclosed
US-5298220-A Forming a coating of a solution containing anioic and cationic dyes and water insoluble organonitrogen compound, drying SHIN-ETSU CHEMICAL CO., LTD. (JP) 1994-03-29 US disclosed
US-5196164-A During addition polymerization, wall coating of anionic dye and cationic dye and organonitrogen compound SHIN-ETSU CHEMICAL CO., LTD. (JP) 1993-03-23 US disclosed
CN-1040206-A Prevent to form the method for polymer scale formation SHINETSU CHEMICAL CO (JP) 1990-03-07 CN disclosed
EP-0355575-A2 Method of preventing polymer scale formation Shin-Etsu Chemical Co., Ltd. (JP) 1990-02-28 EP disclosed
CN-1006386-B PROCESS FOR PRODUCTION OF VINYL CHLORIDE POLYMER SHINETSU CHEM IND CO (JP) 1990-01-10 CN disclosed
EP-0172427-B1 PROCESS FOR PRODUCTION OF VINYL CHLORIDE POLYMER Shin-Etsu Chemical Co., Ltd. (JP) 1989-07-05 EP disclosed
US-4758639-A Process for production of vinyl polymer SHIN-ETSU CHEMICAL CO., LTD. (JP) 1988-07-19 US disclosed
US-4757124-A Suspension or emulsion polymerizing vinyl chloride monomer or mixture of vinyl chloride with vinyl monomer copolymerizable therewith in reactor with walls coated with antiscaling compound containing dye or pigments SHIN-ETSU CHEMICAL CO., LTD. (JP) 1988-07-12 US disclosed
CN-85107531-A Process for producing vinyl chloride polymer 1987-01-21 CN disclosed
EP-0172427-A2 Process for production of vinyl chloride polymer Shin-Etsu Chemical Co., Ltd. (JP) 1986-02-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260103736-A1 Methods Of Improving Production Of Morphinan Alkaloids And Derivatives OPRK1, OPRM1, OPRD1 CYP3A4 13/4885CYP2C9 27/4885CYP2C19 40/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.