SCHEMBL8224196

SCHEMBL8224196

Bc1ccc2c(c1C)CC[C@@H]2NC(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.39
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
KDM1A O60341 2/20 0.37
MAOB P27338 1/20 0.36
EPHX2 P34913 1/20 0.35
DRD2 P14416 3/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
BTK Q06187 1/20 0.34
KCNA3 P22001 1/20 0.34
DRD3 P35462 1/20 0.34
TRPV1 Q8NER1 2/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8185765 0.87 GAA (0.40) GAANFKB1NFKB2RELAKDM1A
SCHEMBL8181064 0.85 GAA (0.39) GAANFKB1NFKB2RELAKDM1A
SCHEMBL8187705 0.85 GAA (0.39) GAANFKB1NFKB2RELAKDM1A
SCHEMBL8181233 0.84 ADAMTS4 (0.39) GAANFKB1NFKB2RELAKDM1A
SCHEMBL10163713 0.84 GAA (0.38) GAANFKB1NFKB2RELAKDM1A
SCHEMBL8183929 0.84 GAA (0.38) GAANFKB1NFKB2RELAKDM1A
SCHEMBL8247296 0.83 GAA (0.37) GAANFKB1NFKB2RELAKDM1A
SCHEMBL4082429 0.83 S1PR1 (0.40) GAANFKB1NFKB2RELAKDM1A
SCHEMBL5429659 0.83 S1PR1 (0.40) GAANFKB1NFKB2RELAKDM1A
SCHEMBL8179948 0.83 GAA (0.37) GAANFKB1NFKB2RELAKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008002671-A2 METALLOPROTEASE INHIBITORS ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2008-01-03 WO disclosed