SCHEMBL8224387

SCHEMBL8224387

Bc1cc2c(O[C@H]3CN[C@H](C(=O)OC)C3)cc(OCC)nc2cc1OC

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.36
PIM1 P11309 1/20 0.36
P2RX3 P56373 1/20 0.34
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
CHEK2 O96017 2/20 0.31
F2 P00734 1/20 0.30
F10 P00742 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7996413 0.87 KDR (0.35) KDRPIM1P2RX3HTR3EHTR3B
Hydrochloric Acid SCHEMBL1071131 0.86 KDR (0.35) KDRPIM1P2RX3HTR3EHTR3B
Hydrochloric Acid SCHEMBL3494749 0.78 STING1 (0.36) HTR3EHTR3BHTR3AHTR3DHTR3C
Hydrochloric Acid SCHEMBL2897201 0.78 STING1 (0.36) HTR3EHTR3BHTR3AHTR3DHTR3C
Hydrochloric Acid SCHEMBL1073116 0.74 PIM1 (0.36) KDRPIM1P2RX3HTR3EHTR3B
SCHEMBL8277445 0.73 PDPK1 (0.34) KDRPIM1HTR3EHTR3BHTR3A
SCHEMBL12963793 0.71 STING1 (0.30) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL12035328 0.69 KDM4E (0.46) KDRPIM1CHEK2
SCHEMBL12335771 0.69 NTSR1 (0.42) PIM1HTR3A
SCHEMBL8222303 0.69 PIM1 (0.41) KDRPIM1CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008057208-A2 HCV NS3 PROTEASE INHIBITORS MERCK & CO., INC. (US) 2008-05-15 WO disclosed