SCHEMBL8224871

SCHEMBL8224871

CC[C@H](C)CNC(=O)N1CCC2(CC1)CN(C)C2c1ccc(F)cc1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 14/20 0.62
NAMPT P43490 2/20 0.42
CYP2C19 P33261 1/20 0.40
FAAH O00519 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
TSHR P16473 1/20 0.38
ALOX12 P18054 1/20 0.38
MAPK1 P28482 1/20 0.38
MTOR P42345 1/20 0.38
RAB9A P51151 1/20 0.38
OPRK1 P41145 1/20 0.38
TACR1 P25103 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8224825 0.89 CACNA1H (0.67) CACNA1HNAMPTCYP2C19FAAHCYP3A4
SCHEMBL8226405 0.88 CACNA1H (0.50) CACNA1HNAMPTCYP2C19FAAHCYP3A4
SCHEMBL8217859 0.87 CACNA1H (0.61) CACNA1HNAMPTCYP2C19OPRK1
SCHEMBL8225775 0.80 CACNA1H (0.83) CACNA1H
SCHEMBL8224691 0.79 CACNA1H (0.54) CACNA1HNAMPT
SCHEMBL13595952 0.77 CACNA1H (0.70) CACNA1H
SCHEMBL13595944 0.77 CACNA1H (1.00) CACNA1HCYP2C19CYP2D6TSHR
SCHEMBL13596146 0.76 CACNA1H (0.65) CACNA1H
SCHEMBL13595951 0.74 CACNA1H (0.79) CACNA1HCYP2D6RAB9A
SCHEMBL8218861 0.73 CACNA1H (0.70) CACNA1HCYP2C19TSHRRAB9AOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033456-A1 SPIRO-CONDENSED AZETIDINE DERIVATIVES USEFUL IN TREATING PAIN, DIABETES AND DISORDERS OF LIPID METABILISM SCHERING CORPORATION (US) 2008-03-20 WO disclosed