SCHEMBL8224825

SCHEMBL8224825

CC[C@H](C)CNC(=O)N1CCC2(CC1)CN(C(C)C)C2c1ccc(F)cc1

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 15/20 0.67
NAMPT P43490 1/20 0.39
CYP2C19 P33261 1/20 0.39
HRH3 Q9Y5N1 1/20 0.36
S1PR2 O95136 1/20 0.36
FAAH O00519 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
ALOX12 P18054 1/20 0.35
MAPK1 P28482 1/20 0.35
MTOR P42345 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8224691 0.90 CACNA1H (0.54) CACNA1HNAMPT
SCHEMBL8224871 0.89 CACNA1H (0.62) CACNA1HNAMPTCYP2C19FAAHCYP3A4
SCHEMBL8217859 0.86 CACNA1H (0.61) CACNA1HNAMPTCYP2C19
SCHEMBL8226405 0.85 CACNA1H (0.50) CACNA1HNAMPTCYP2C19FAAHCYP3A4
SCHEMBL8219197 0.84 CACNA1H (0.78) CACNA1H
SCHEMBL8224684 0.80 CACNA1H (1.00) CACNA1H
SCHEMBL8218859 0.80 CACNA1H (1.00) CACNA1HCYP2C19S1PR2CYP2D6
SCHEMBL13595981 0.78 CACNA1H (0.84) CACNA1H
SCHEMBL8225905 0.78 CACNA1H (0.78) CACNA1H
SCHEMBL13595938 0.77 CACNA1H (0.84) CACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008033456-A1 SPIRO-CONDENSED AZETIDINE DERIVATIVES USEFUL IN TREATING PAIN, DIABETES AND DISORDERS OF LIPID METABILISM SCHERING CORPORATION (US) 2008-03-20 WO disclosed