SCHEMBL8225952

SCHEMBL8225952

O=C1CCN2C(=O)c3ccccc3OC2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.41
ADORA3 P0DMS8 3/20 0.40
AR P10275 2/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP19A1 P11511 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GRIA1 P42261 1/20 0.37
CDK5 Q00535 1/20 0.37
DYRK1A Q13627 1/20 0.37
CDK5R1 Q15078 1/20 0.37
SIGMAR1 Q99720 2/20 0.36
ABCB1 P08183 1/20 0.36
HSD11B1 P28845 1/20 0.35
AKR1C3 P42330 1/20 0.35
NPC1 O15118 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
KDM1A O60341 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31562964 0.81 GRIA1 (0.47) MAOBADORA3ARKDM4ECYP19A1
SCHEMBL8216824 0.80 TUBB4A (0.47) MAOBARCYP19A1GRIA1MAPT
SCHEMBL31563001 0.78 GRIA1 (0.58) MAOBADORA3ARKDM4ECYP19A1
SCHEMBL31562979 0.76 PARP1 (0.43) MAOBADORA3ARKDM4ECYP19A1
SCHEMBL5618588 0.75 HTR2C (0.55) HTR2CHTR2BHTR2A
SCHEMBL5619702 0.75 HTR2C (0.55) HTR2CHTR2BHTR2A
SCHEMBL5618115 0.75 HTR2C (0.55) HTR2CHTR2BHTR2A
SCHEMBL7377181 0.69
SCHEMBL31562965 0.68 HSD17B10 (0.38) MAOBADORA3ARKDM4ECYP19A1
SCHEMBL31562958 0.67 AR (0.36) MAOBADORA3ARKDM4ECYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000006576-A1 COMPOUNDS ASTRAZENECA AB (SE) 2000-02-10 WO disclosed