SCHEMBL8230204

SCHEMBL8230204

C=CCCCCN[C@H](C(=O)N1C[C@H](OCc2cccc(-c3cccc(/C=C\C)c3)c2)C[C@H]1C(=O)OC)C1CCCCC1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.34
CYP3A4 P08684 1/20 0.33
THRB P10828 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MMP2 P08253 2/20 0.31
ANPEP P15144 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MC4R P32245 1/20 0.30
MC3R P41968 1/20 0.30
MC1R Q01726 1/20 0.30
AGTR2 P50052 1/20 0.30
NR1H4 Q96RI1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2427392 0.94 F2 (0.35) F2CYP3A4THRBHSD17B10MMP2
SCHEMBL4303372 0.87 AGTR2 (0.36) F2CYP3A4THRBHSD17B10MC4R
SCHEMBL2429307 0.81 ABCB1 (0.34) MMP2ANPEPMC4RMC3RMC1R
SCHEMBL2426240 0.79 KLK5 (0.40) F2CYP3A4THRBHSD17B10
SCHEMBL8228152 0.79 CYP3A4 (0.38) CYP3A4THRBHSD17B10MMP2MC4R
Hydrochloric Acid SCHEMBL2429662 0.78 CYP3A4 (0.38) F2CYP3A4THRBHSD17B10MMP2
SCHEMBL2431251 0.77 ABCB1 (0.34) MC4RMC3RMC1RAGTR2
SCHEMBL2427394 0.76 CYP3A4 (0.34) F2CYP3A4THRBHSD17B10
SCHEMBL4294862 0.73 ACE (0.40) F2CYP3A4THRBHSD17B10AGTR2
SCHEMBL2430508 0.72 CACNA1B (0.41) CYP3A4THRBHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007148135-A1 MACROCYCLIC COMPOUNDS AS ANTIVIRAL AGENTS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2007-12-27 WO disclosed