SCHEMBL8230449

SCHEMBL8230449

Bc1cc(C(=O)NCC2CCN(CC3CCOCC3)CC2)c2c(c1N)CCCO2

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 15/20 0.49
ACHE P22303 2/20 0.43
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2332701 0.89 HTR4 (0.51) HTR4ACHECYP3A4CYP2D6
Hydrochloric Acid SCHEMBL5631883 0.89 HTR4 (0.50) HTR4ACHECYP3A4CYP2D6
Succinic Acid SCHEMBL5632076 0.85 HTR4 (0.47) HTR4ACHECYP3A4CYP2D6
SCHEMBL2331750 0.84 HTR4 (0.53) HTR4ACHEHTR3EHTR3BHTR3A
SCHEMBL2333431 0.84 HTR4 (0.53) HTR4ACHEHTR3EHTR3BHTR3A
SCHEMBL2331760 0.84 HTR4 (0.53) HTR4ACHEHTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL5332277 0.83 HTR4 (0.47) HTR4ACHEHTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL5316450 0.83 HTR4 (0.53) HTR4ACHEHTR3EHTR3BHTR3A
SCHEMBL5630511 0.80 HTR4 (0.45) HTR4ACHECYP3A4CYP2D6MEN1
SCHEMBL2329530 0.79 HTR4 (0.51) HTR4ACHEALDH1A1HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096352-A1 5-AMINO-6-BROMO-N-{ [1- (TETRAHYDR0-2H-PYRAN-4-YLMETHYL) -4-PIPERIDINYL] METHYL}-3, 4 -DIHYDRO-2H-CHROMENE-8-CARBOXAMIDE AS 5-HT4 RECEPTOR AGONIST GLAXO GROUP LIMITED (GB) 2007-08-30 WO disclosed