SCHEMBL8230626

SCHEMBL8230626

NOC1CCc2ccccc2C1

nearest known ligand 0.72

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 7/20 0.72
PLAU P00749 1/20 0.55
ANPEP P15144 2/20 0.47
HTR2C P28335 1/20 0.47
SLC6A4 P31645 1/20 0.47
HTR2B P41595 1/20 0.47
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
GRIN2B Q13224 1/20 0.40
HTR1A P08908 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3087762 0.84 IDO1 (1.00) IDO1PLAUANPEPCA1CA2
SCHEMBL11852553 0.83 PLAU (0.54) IDO1PLAUANPEPHTR2CSLC6A4
SCHEMBL6570375 0.79 CYP1A2 (0.51) IDO1PLAUANPEPHTR2CSLC6A4
SCHEMBL6311069 0.79 CYP1A2 (0.51) IDO1PLAUANPEPHTR2CSLC6A4
SCHEMBL22524385 0.79 CYP1A2 (0.51) IDO1PLAUANPEPHTR2CSLC6A4
SCHEMBL13456262 0.76 PLAU (0.47) IDO1PLAUANPEPHTR2CSLC6A4
SCHEMBL11555929 0.75 PLAU (0.46) IDO1PLAUANPEPHTR2CSLC6A4
SCHEMBL10447404 0.75 CYP1A2 (0.55) IDO1PLAUANPEPHTR2CSLC6A4
SCHEMBL8530045 0.74 IDO1 (0.44) IDO1PLAUANPEPHTR2CSLC6A4
SCHEMBL26944395 0.73 IDO1 (0.43) IDO1PLAUANPEPHTR2CSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2032585-B1 SUBSTITUTED PTERIDINES AS THERAPEUTIC AGENTS BOEHRINGER INGELHEIM INT (DE) 2014-07-23 EP disclosed
WO-2007135026-A2 SUBSTITUTED PTERIDINES AS THERAPEUTIC AGENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-11-29 WO disclosed