SCHEMBL8235141

SCHEMBL8235141

CCn1c(N2CCO[C@H]3c4ccccc4CC[C@H]32)nc(-c2ccncc2)cc1=O

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 14/20 0.44
CYP1A2 P05177 3/20 0.44
CYP2D6 P10635 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL697318 0.89 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL697319 0.89 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL8234283 0.89 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL698081 0.89 GSK3B (0.55) GSK3BCYP1A2CYP2D6
SCHEMBL8227103 0.81 GSK3B (0.46) GSK3BCYP1A2CYP2D6
SCHEMBL8232107 0.79 GSK3B (0.56) GSK3BCYP1A2CYP2D6
SCHEMBL696848 0.79 GSK3B (0.54) GSK3BCYP1A2CYP2D6
SCHEMBL696849 0.79 GSK3B (0.54) GSK3BCYP1A2CYP2D6
SCHEMBL698095 0.79 GSK3B (0.54) GSK3BCYP1A2CYP2D6
SCHEMBL8232077 0.79 GSK3B (0.54) GSK3BCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007119463-A1 2-(CYCLIC AMINO)-PYRIMIDONE DERIVATIVES AS TPK1 INHIBITORS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-10-25 WO disclosed