SCHEMBL8235283

SCHEMBL8235283

CCn1c(N2CCC[C@H]2C(N)=O)nc(-c2ccncc2)cc1=O

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 14/20 0.42
KDM1A O60341 1/20 0.40
CYP1A2 P05177 3/20 0.39
CYP2D6 P10635 3/20 0.39
ELANE P08246 2/20 0.38
AADAT Q8N5Z0 2/20 0.36
CDC7 O00311 1/20 0.36
ROCK2 O75116 1/20 0.36
PIM1 P11309 1/20 0.36
HIPK2 Q9H2X6 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13711423 0.86 GSK3B (0.57) GSK3BCYP1A2CYP2D6
SCHEMBL696646 0.82 GSK3B (0.47) GSK3BKDM1ACYP1A2CYP2D6
SCHEMBL8227103 0.76 GSK3B (0.46) GSK3BKDM1ACYP1A2CYP2D6
SCHEMBL8235423 0.76 GSK3B (0.41) GSK3BCYP1A2CYP2D6CDC7ROCK2
SCHEMBL8234209 0.74 GSK3B (0.48) GSK3BKDM1ACYP1A2CYP2D6
SCHEMBL8232926 0.74 GSK3B (0.48) GSK3BKDM1ACYP1A2CYP2D6
SCHEMBL13711424 0.73 GSK3B (0.60) GSK3BCYP1A2CYP2D6
SCHEMBL8231807 0.73 GSK3B (0.51) GSK3BCYP1A2CYP2D6
SCHEMBL696647 0.73 GSK3B (0.41) GSK3BKDM1ACYP1A2CYP2D6
SCHEMBL8235150 0.71 GSK3B (0.51) GSK3BCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007119463-A1 2-(CYCLIC AMINO)-PYRIMIDONE DERIVATIVES AS TPK1 INHIBITORS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-10-25 WO disclosed