SCHEMBL696646

SCHEMBL696646

CCn1c(N2CCCC3CCCCC32)nc(-c2ccncc2)cc1=O

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 17/20 0.47
CYP1A2 P05177 3/20 0.40
CYP2D6 P10635 3/20 0.40
KDM1A O60341 1/20 0.40
LATS1 O95835 1/20 0.39
MAPK13 O15264 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8227103 0.87 GSK3B (0.46) GSK3BCYP1A2CYP2D6KDM1A
SCHEMBL696622 0.85 GSK3B (0.60) GSK3BCYP1A2CYP2D6
SCHEMBL8234773 0.85 GSK3B (0.60) GSK3BCYP1A2CYP2D6
SCHEMBL8235283 0.82 GSK3B (0.42) GSK3BCYP1A2CYP2D6KDM1A
SCHEMBL8232926 0.77 GSK3B (0.48) GSK3BCYP1A2CYP2D6KDM1A
SCHEMBL8234209 0.77 GSK3B (0.48) GSK3BCYP1A2CYP2D6KDM1A
SCHEMBL8231807 0.75 GSK3B (0.51) GSK3BCYP1A2CYP2D6
SCHEMBL696647 0.75 GSK3B (0.41) GSK3BCYP1A2CYP2D6KDM1A
SCHEMBL8235141 0.75 GSK3B (0.44) GSK3BCYP1A2CYP2D6
SCHEMBL696934 0.74 GSK3B (0.57) GSK3BCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423207-A2 2-(cyclic amino)-pyrimidone derivatives as TPK1 inhibitors Mitsubishi Tanabe Pharma Corporation (JP) 2012-02-29 EP disclosed