SCHEMBL8235476

SCHEMBL8235476

CC1=C(c2ccc(NC(=O)c3ccncc3C)cc2)CN(c2ccccn2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.44
KDM4E B2RXH2 7/20 0.44
SMN1; SMN2 Q16637 5/20 0.44
RCE1 Q9Y256 2/20 0.44
TRPV1 Q8NER1 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
MAPT P10636 6/20 0.43
CYP1A2 P05177 1/20 0.43
GAA P10253 3/20 0.42
NAMPT P43490 1/20 0.42
TYK2 P29597 1/20 0.41
PANK3 Q9H999 1/20 0.39
HTT P42858 2/20 0.39
SLC11A2 P49281 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MAPK1 P28482 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL615223 0.91 KDM4E (0.43) ALDH1A1KDM4ESMN1; SMN2RCE1TRPV1
SCHEMBL12603918 0.85 MAPT (0.47) ALDH1A1KDM4ESMN1; SMN2RCE1TRPV1
SCHEMBL1780945 0.85 TRPV1 (0.47) ALDH1A1SMN1; SMN2TRPV1L3MBTL1GAA
SCHEMBL1783971 0.84 TRPV1 (0.45) ALDH1A1KDM4ESMN1; SMN2RCE1TRPV1
SCHEMBL8228702 0.84 PDGFRB (0.39) ALDH1A1KDM4ESMN1; SMN2L3MBTL1MAPT
SCHEMBL989336 0.83 TRPV1 (0.44) ALDH1A1KDM4ESMN1; SMN2TRPV1L3MBTL1
SCHEMBL7920420 0.83 TRPV1 (0.44) ALDH1A1KDM4ESMN1; SMN2RCE1TRPV1
SCHEMBL8232016 0.83 CYP1A2 (0.36) ALDH1A1KDM4ESMN1; SMN2L3MBTL1MAPT
Hydrochloric Acid SCHEMBL1782050 0.83 TRPV1 (0.44) ALDH1A1KDM4ESMN1; SMN2RCE1TRPV1
SCHEMBL1780548 0.83 MAPT (0.39) ALDH1A1KDM4ESMN1; SMN2TRPV1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007087443-A2 VINYL-PHENYL DERIVATIVES FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2007-08-02 WO disclosed