SCHEMBL8236221

SCHEMBL8236221

Cc1ccc(-c2ncco2)cc1-c1ccc(NC(=O)c2c(C)cccc2F)cn1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IL2 P60568 17/20 0.61
STIM1 Q13586 1/20 0.42
ORAI1 Q96D31 1/20 0.42
ORAI2 Q96SN7 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
GRM1 Q13255 1/20 0.40
GRM4 Q14833 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2812970 0.96 IL2 (0.66) IL2STIM1ORAI1NPC1RAB9A
Hydrochloric Acid SCHEMBL2811428 0.95 IL2 (0.65) IL2STIM1ORAI1NPC1RAB9A
SCHEMBL8261671 0.90 IL2 (0.66) IL2STIM1ORAI1
SCHEMBL4762567 0.86 IL2 (0.71) IL2STIM1ORAI1
SCHEMBL2812935 0.85 IL2 (0.54) IL2NPC1RAB9A
Hydrochloric Acid SCHEMBL2813897 0.84 IL2 (0.53) IL2NPC1RAB9A
SCHEMBL5554286 0.83 IL2 (0.69) IL2STIM1ORAI1ORAI2
SCHEMBL2814805 0.83 IL2 (0.53) IL2NPC1RAB9A
SCHEMBL2813970 0.82 CYP11B2 (0.47) IL2NPC1RAB9A
SCHEMBL2813079 0.80 IL2 (0.44) IL2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007089904-A2 PYRIDYLPHENYL COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2007-08-09 WO disclosed