SCHEMBL8237694

SCHEMBL8237694

CCCCCN1C(=O)C(C)(C)Oc2ccc(N(C(=O)[C@H]3CNC[C@@H](C(=O)NC(C)(C)c4ccccc4)C3)C3CC3)cc21

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
REN P00797 3/20 0.46
SCN9A Q15858 6/20 0.36
ALDH1A1 P00352 2/20 0.34
SSTR4 P31391 1/20 0.33
GAA P10253 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TSHR P16473 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL89616 0.92 REN (0.53) RENALDH1A1TDP1CYP1A2CYP2C9
SCHEMBL90241 0.91 REN (0.49) RENALDH1A1SSTR4GAATDP1
SCHEMBL8229861 0.87 REN (0.36) RENSCN9AALDH1A1TDP1CYP1A2
SCHEMBL89679 0.85 REN (0.47) RENALDH1A1SSTR4TDP1CYP1A2
SCHEMBL90208 0.84 REN (0.56) RENTDP1CYP1A2CYP2C9CYP2C19
SCHEMBL8235471 0.84 REN (0.56) RENTDP1CYP1A2CYP2C9CYP2C19
SCHEMBL90491 0.83 REN (0.46) RENALDH1A1TDP1CYP1A2CYP2C9
SCHEMBL8238499 0.82 REN (0.59) RENALDH1A1MEN1KMT2A
SCHEMBL8235599 0.82 REN (0.45) RENSCN9AALDH1A1GAAMEN1
SCHEMBL8238346 0.82 REN (0.54) RENALDH1A1GAATDP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007077005-A1 3 , 5-SUBSTITΓUED PIPERIDINE COMPOUNDS AS RENIN INHIBITORS NOVARTIS AG (CH) 2007-07-12 WO disclosed