SCHEMBL8239271

SCHEMBL8239271

Nc1ccc(N2CCN(C(=O)C3CCCO3)CC2)cc1

nearest known ligand 0.71

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.71
NAMPT P43490 1/20 0.60
KDM4E B2RXH2 2/20 0.59
TSHR P16473 2/20 0.59
HSD17B10 Q99714 1/20 0.59
HTT P42858 1/20 0.57
CASP6 P55212 1/20 0.52
GFER P55789 1/20 0.52
FASN P49327 2/20 0.52
PKM P14618 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
POLB P06746 1/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HPGD P15428 1/20 0.49
LMNA P02545 1/20 0.49
GLA P06280 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3636273 0.82 NAMPT (0.61) ALDH1A1NAMPTKDM4ETSHRHSD17B10
SCHEMBL14963886 0.82 HPGD (0.71) ALDH1A1NAMPTHTTPOLBMEN1
SCHEMBL189163 0.79 ALDH1A1 (0.69) ALDH1A1NAMPTKDM4ETSHRHSD17B10
SCHEMBL1663638 0.78 TDP1 (0.73) ALDH1A1NAMPTKDM4EHSD17B10HTT
SCHEMBL3216413 0.76 TDP1 (0.66) ALDH1A1NAMPTKDM4EHSD17B10HTT
SCHEMBL12156680 0.76 ALDH1A1 (0.52) ALDH1A1KDM4ETSHRHSD17B10HTT
SCHEMBL3706326 0.76 NAMPT (1.00) NAMPT
Hydrochloric Acid SCHEMBL3205122 0.75 TDP1 (0.64) ALDH1A1NAMPTKDM4EHSD17B10HTT
SCHEMBL3209251 0.74 KMT2A (0.59) ALDH1A1NAMPTKDM4ETSHRHSD17B10
SCHEMBL28312550 0.74 RECQL (0.63) ALDH1A1KDM4ETSHRHSD17B10HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007089768-A2 4-ARYL-2-AMINO-PYRIMIDINES OR 4-ARYL-2-AMINOALKYL-PYRIMIDINES AS JAK-2 MODULATORS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM EXELIXIS, INC. (US) 2007-08-09 WO disclosed