SCHEMBL8239387

SCHEMBL8239387

CSc1ccccc1-c1ccc(-c2csc(C)n2)cn1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.43
KDM4E B2RXH2 3/20 0.43
POLB P06746 2/20 0.43
RAB9A P51151 2/20 0.43
HTT P42858 1/20 0.43
TGFBR1 P36897 1/20 0.42
MAPT P10636 2/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
HPGD P15428 2/20 0.41
ALDH1A1 P00352 1/20 0.41
RECQL P46063 1/20 0.41
ESR2 Q92731 1/20 0.41
NPC1 O15118 1/20 0.41
STAT1 P42224 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8240041 0.86 RECQL (0.40) GAAKDM4EPOLBRAB9AHTT
SCHEMBL8242243 0.85 KDM4E (0.49) GAAKDM4EPOLBRAB9AHTT
SCHEMBL11982656 0.82 KDM4E (0.46) GAAKDM4EPOLBRAB9AHTT
SCHEMBL8239502 0.82 MPL (0.51) GAAKDM4EPOLBRAB9AHTT
SCHEMBL11982667 0.81 RAB9A (0.52) GAAKDM4EPOLBRAB9AHTT
SCHEMBL11982626 0.80 MAPT (0.51) GAAMAPTRECQL
SCHEMBL11982627 0.80 RECQL (0.44) GAAKDM4EPOLBRAB9AHTT
SCHEMBL8239608 0.79 RAB9A (0.47) GAAKDM4EPOLBRAB9AHTT
SCHEMBL11982625 0.79 GAA (0.52) GAAKDM4ETGFBR1
SCHEMBL8238546 0.77 RECQL (0.43) GAAKDM4EPOLBRAB9AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007050050-A2 THIAZOLYL MGLUR5 ANTAGONISTS AND METHODS FOR THEIR USE MERCK & CO., INC. (US) 2007-05-03 WO disclosed