SCHEMBL8239887

SCHEMBL8239887

C=C(Nc1cc(-c2cccs2)ccc1N)c1ccc(-c2ccc3c(c2)NC(=O)[C@H](Cc2c[nH]c4ccccc24)N3)cc1

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 15/20 0.45
HDAC2 Q92769 9/20 0.45
HDAC3 O15379 7/20 0.45
GSK3B P49841 2/20 0.39
IDO1 P14902 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5137947 0.92 HDAC1 (0.53) HDAC1HDAC2HDAC3
SCHEMBL5075712 0.92 HDAC1 (0.53) HDAC1HDAC2HDAC3
SCHEMBL5579382 0.74 HDAC3 (0.53) HDAC1HDAC2HDAC3GSK3BIDO1
SCHEMBL5579378 0.74 HDAC3 (0.53) HDAC1HDAC2HDAC3GSK3BIDO1
SCHEMBL5079028 0.69 IDO1 (0.55) HDAC1HDAC2HDAC3GSK3BIDO1
SCHEMBL5082100 0.69 IDO1 (0.55) HDAC1HDAC2HDAC3GSK3BIDO1
SCHEMBL6038011 0.67 GSK3B (0.72) GSK3BIDO1
SCHEMBL6038005 0.67 GSK3B (0.72) GSK3BIDO1
SCHEMBL5579406 0.67 IDO1 (0.61) GSK3BIDO1
SCHEMBL5579410 0.67 IDO1 (0.61) GSK3BIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007022638-A1 BENZODIAZEPINE AND BENZOPIPERAZINE ANALOG INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2007-03-01 WO disclosed