SCHEMBL8240

SCHEMBL8240

O=C(O)c1cc2ccc(-c3nnn[nH]3)cc2n1O

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LDHA P00338 7/20 0.58
DAO P14920 1/20 0.47
CCR2 P41597 2/20 0.33
MCL1 Q07820 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7982 0.76 LDHA (0.58) LDHADAOALDH1A1
SCHEMBL14118756 0.74 LDHA (0.56) LDHADAOALDH1A1
SCHEMBL7814 0.74 LDHA (1.00) LDHADAOCCR2MCL1ALDH1A1
SCHEMBL7300 0.74 LDHA (1.00) LDHADAOCCR2MCL1ALDH1A1
SCHEMBL13306 0.73 LDHA (0.79) LDHADAOCCR2
SCHEMBL7108 0.72 LDHA (0.82) LDHADAOCCR2MCL1ALDH1A1
SCHEMBL7835 0.72 LDHA (0.77) LDHADAOCCR2MCL1
SCHEMBL7582 0.72 LDHA (0.77) LDHADAOCCR2MCL1ALDH1A1
SCHEMBL8712 0.70 LDHA (0.78) LDHADAOCCR2ALDH1A1
SCHEMBL2761565 0.69 MCL1 (0.51) MCL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499114-A1 COMPOUNDS INHIBITORS OF ENZYME LACTATE DEHYDROGENASE (LDH) AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS Universita Di Pisa (IT) 2012-09-19 EP disclosed
WO-2011054525-A1 COMPOUNDS INHIBITORS OF ENZYME LACTATE DEHYDROGENASE (LDH) AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS UNIVERSITA' DI PISA (IT) 2011-05-12 WO disclosed