SCHEMBL8240482

SCHEMBL8240482

O=C(NCc1cc(Cl)ccc1F)NC(c1ccccc1)c1nc(-c2ccc3[nH]c(=O)cc(O)c3c2)c(Cl)[nH]1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
F11 P03951 11/20 0.43
ROCK2 O75116 3/20 0.39
KLKB1 P03952 2/20 0.38
UBASH3B Q8TF42 1/20 0.36
MAPK3 P27361 1/20 0.35
MAPK1 P28482 1/20 0.35
PRSS1 P07477 2/20 0.34
PRSS2 P07478 2/20 0.34
PRSS3 P35030 2/20 0.34
TRPV1 Q8NER1 2/20 0.34
ROCK1 Q13464 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1198076 0.88 F11 (0.53) F11ROCK2KLKB1PRSS1PRSS2
SCHEMBL1198074 0.88 F11 (0.53) F11ROCK2KLKB1PRSS1PRSS2
SCHEMBL1195928 0.82 F11 (0.49) F11ROCK2KLKB1PRSS1PRSS2
SCHEMBL13387419 0.81 F11 (0.40) F11KLKB1UBASH3BTRPV1
SCHEMBL13387420 0.79 F11 (0.39) F11KLKB1UBASH3BMAPK1TRPV1
SCHEMBL13552343 0.79 F11 (0.43) F11ROCK2KLKB1PRSS1PRSS2
SCHEMBL1196691 0.77 F11 (0.50) F11KLKB1PRSS1PRSS2PRSS3
SCHEMBL1196693 0.77 F11 (0.50) F11KLKB1PRSS1PRSS2PRSS3
SCHEMBL1196558 0.77 F11 (0.65) F11KLKB1PRSS1PRSS2PRSS3
SCHEMBL1196556 0.77 F11 (0.65) F11KLKB1PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007070826-A1 ARYLPROPIONAMIDE, ARYLACRYLAMIDE, ARYLPROPYNAMIDE, OR ARYLMETHYLUREA ANALOGS AS FACTOR XIA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-06-21 WO disclosed