SCHEMBL8243722

SCHEMBL8243722

O=C(CCn1ccc2cc(Cl)ccc21)N1CCC(S(=O)(=O)NC2=CC=CCC2)C1

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.38
KRAS P01116 2/20 0.37
NPY5R Q15761 1/20 0.35
F10 P00742 6/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
KMO O15229 1/20 0.35
ACLY P53396 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL66061 0.83 HRH3 (0.41) HRH3KRASNPY5RF10TP53
SCHEMBL57307 0.79 HRH3 (0.48) HRH3KRASF10TP53MAPT
SCHEMBL65671 0.78 F10 (0.44) HRH3KRASNPY5RF10TP53
SCHEMBL57175 0.77 TACR1 (0.43) HRH3KRASNPY5RF10TP53
SCHEMBL56764 0.74 F10 (0.44) HRH3KRASNPY5RF10MAPT
SCHEMBL66257 0.74 F2 (0.43) HRH3NPY5RF10TP53MAPT
SCHEMBL8242528 0.72 MEN1 (0.50) HRH3KRASF10TP53MAPT
SCHEMBL8243869 0.67 SMN1; SMN2 (0.43) MAPT
SCHEMBL1576317 0.65 SCN9A (0.44) F10
SCHEMBL10310789 0.65 F10 (0.44) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007050522-A1 DERIVATIVES FOR MODULATION OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-05-03 WO disclosed