SCHEMBL8245208

SCHEMBL8245208

O=C(O)c1nc2ccnn2c2c1CCN2C1CCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.39
HTR2A P28223 4/20 0.36
HTR2B P41595 4/20 0.36
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
MAPK1 P28482 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
PDE4B Q07343 7/20 0.33
PDE4D Q08499 7/20 0.33
RAD52 P43351 1/20 0.33
ACVR1 Q04771 1/20 0.32
PDE4A P27815 5/20 0.31
PDE4C Q08493 5/20 0.31
CCNT1 O60563 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8177219 0.98 HTR2C (0.39) HTR2CHTR2AHTR2BKMT2AKDM4E
SCHEMBL8177229 0.84 KMT2A (0.40) HTR2CHTR2AHTR2BKMT2AKDM4E
SCHEMBL8191337 0.84 PDE4A (0.47) HTR2CKMT2AKDM4EALDH1A1POLB
SCHEMBL8189529 0.83 KMT2A (0.39) HTR2CHTR2AHTR2BKMT2AKDM4E
SCHEMBL8187166 0.82 HTR2C (0.36) HTR2CHTR2AHTR2BKMT2AKDM4E
SCHEMBL8187118 0.82 PDE4A (0.47) HTR2CKMT2AKDM4EALDH1A1POLB
SCHEMBL8186875 0.81 KMT2A (0.36) HTR2CHTR2AHTR2BKMT2AKDM4E
SCHEMBL8192426 0.81 PDE4A (0.46) HTR2CKMT2AALDH1A1POLBMAPT
SCHEMBL8176828 0.80 HTR2C (0.41) HTR2CHTR2AHTR2BKMT2AKDM4E
SCHEMBL8191382 0.79 PDE4A (0.48) HTR2CKMT2AKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1021447-A1 PYRROLOPYRAZOLOPYRIMIDINE COMPOUND AND MEDICINE COMPRISING THE SAME POLA CHEMICAL INDUSTRIES, INC. (JP) 2000-07-26 EP disclosed
WO-1998033799-A1 PYRROLOPYRAZOLOPYRIMIDINE COMPOUND AND MEDICINE COMPRISING THE SAME POLA CHEMICAL INDUSTRIES, INC. (JP) 1998-08-06 WO disclosed