SCHEMBL8245688

SCHEMBL8245688

CC1(C)CCc2nc(-c3cn(-c4cc(-c5cccnc5)nc(C5C=CC=CC5)c4)cn3)ccc2C1=O

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.33
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
CYP2E1 P05181 2/20 0.31
CYP2A6 P11509 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2B6 P20813 2/20 0.31
CYP2C19 P33261 2/20 0.31
RIPK2 O43353 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4680870 0.87 GRM5 (0.41) GRM5HSP90AA1HSP90AB1CYP2E1CYP2A6
SCHEMBL4683613 0.83 GRM5 (0.37) GRM5HSP90AA1HSP90AB1CYP2E1CYP2A6
SCHEMBL4740959 0.81 GRM5 (0.46) GRM5
SCHEMBL4737979 0.77 GRM5 (0.38) GRM5HSP90AA1HSP90AB1
SCHEMBL4686025 0.75 GRM5 (0.40) GRM5HSP90AA1HSP90AB1CYP2E1CYP2A6
SCHEMBL6103021 0.75 GRM5 (0.40) GRM5
SCHEMBL13706965 0.74 GRM5 (0.49) GRM5HSP90AA1HSP90AB1CYP2A6CYP2C19
SCHEMBL4683032 0.72 CYP19A1 (0.40) GRM5HSP90AA1HSP90AB1CYP2E1CYP2A6
SCHEMBL4680906 0.72 ALDH1A1 (0.41) GRM5CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL4686152 0.71 GRM5 (0.36) GRM5HSP90AA1CYP2E1CYP2A6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007023245-A1 TETRAHYDROQUINOLINONES AND THEIR USE AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS MERZ PHARMA GMBH & CO. KGAA (DE) 2007-03-01 WO disclosed