SCHEMBL8247149

SCHEMBL8247149

O=C(O)CNC(=O)c1c(O)c2c(O)cccc2n(Cc2ccccc2)c1=O

nearest known ligand 0.73

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 8/20 0.73
EGLN3 Q9H6Z9 6/20 0.62
EGLN2 Q96KS0 2/20 0.51
HIF1A Q16665 1/20 0.51
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
KCNH2 Q12809 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8247310 0.89 EGLN1 (0.61) EGLN1EGLN3EGLN2HIF1AKDM4E
SCHEMBL8238459 0.86 EGLN1 (0.67) EGLN1EGLN3EGLN2HIF1AKDM4E
SCHEMBL5428652 0.85 EGLN1 (0.66) EGLN1EGLN3EGLN2HIF1AKDM4E
SCHEMBL8244419 0.85 EGLN1 (1.00) EGLN1EGLN3EGLN2HIF1AKDM4E
SCHEMBL8248294 0.82 EGLN1 (0.77) EGLN1EGLN3EGLN2HIF1AKDM4E
SCHEMBL5307125 0.80 EGLN1 (0.61) EGLN1EGLN3EGLN2HIF1AKDM4E
SCHEMBL1960754 0.80 EGLN1 (0.71) EGLN1EGLN3EGLN2KDM4EKCNH2
SCHEMBL8247257 0.79 EGLN1 (0.60) EGLN1EGLN3EGLN2HIF1AKDM4E
SCHEMBL8245588 0.79 EGLN1 (0.83) EGLN1EGLN3EGLN2HIF1AKDM4E
SCHEMBL4142379 0.79 KCNH2 (0.74) EGLN1EGLN3EGLN2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007038571-A2 PROLYL HYDROXYLASE ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-05 WO disclosed