SCHEMBL8248281

SCHEMBL8248281

C=C(c1c[nH]c2cc(Cl)ccc12)N1CCC2(CC1)OC(=O)c1ccccc12

nearest known ligand 0.81

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 10/20 0.81
OXTR P30559 1/20 0.56
NPY5R Q15761 7/20 0.52
HSD11B1 P28845 2/20 0.47
CYP2D6 P10635 1/20 0.47
DGAT1 O75907 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4355499 0.89 AVPR1A (1.00) AVPR1AOXTRNPY5RHSD11B1CYP2D6
SCHEMBL8242341 0.89 AVPR1A (0.65) AVPR1AOXTRNPY5RDGAT1
SCHEMBL4364065 0.82 AVPR1A (0.87) AVPR1AOXTRNPY5RHSD11B1CYP2D6
SCHEMBL4355431 0.79 AVPR1A (0.80) AVPR1AOXTRNPY5R
SCHEMBL4357247 0.79 AVPR1A (0.80) AVPR1AOXTRNPY5R
SCHEMBL5138467 0.79 AVPR1A (0.80) AVPR1AOXTRNPY5R
SCHEMBL13602796 0.77 AVPR1A (0.78) AVPR1AOXTRNPY5R
SCHEMBL8248461 0.77 AVPR1A (0.49) AVPR1AOXTRHSD11B1
SCHEMBL4365900 0.77 AVPR1A (0.76) AVPR1AOXTR
SCHEMBL4759170 0.76 AVPR1A (1.00) AVPR1AOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007006688-A1 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO disclosed