SCHEMBL8248461

SCHEMBL8248461

C=C(c1c[nH]c2cc(Cl)ccc12)N1CCC2(C=Cc3ccccc32)CC1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 11/20 0.49
HSD11B1 P28845 1/20 0.49
OXTR P30559 1/20 0.48
MCHR2 Q969V1 1/20 0.40
SSTR2 P30874 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4363635 0.88 AVPR1A (0.64) AVPR1AHSD11B1OXTRMCHR2
SCHEMBL8248281 0.77 AVPR1A (0.81) AVPR1AHSD11B1OXTR
SCHEMBL14609348 0.76 DRD3 (0.47) AVPR1AOXTR
SCHEMBL12024234 0.75 DRD2 (0.47) AVPR1AOXTR
SCHEMBL14609342 0.74 AVPR1A (0.43) AVPR1AOXTR
SCHEMBL14609585 0.74 AVPR1A (0.57) AVPR1AOXTR
SCHEMBL12024671 0.72 AVPR1A (0.76) AVPR1AHSD11B1OXTR
SCHEMBL12024705 0.72 DRD2 (0.43) AVPR1AOXTR
SCHEMBL8242341 0.70 AVPR1A (0.65) AVPR1AOXTR
SCHEMBL13971036 0.69 HSD11B1 (0.48) HSD11B1OXTRMCHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007006688-A1 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO disclosed