SCHEMBL8250426

SCHEMBL8250426

Cc1cccc(N=C2C(=O)N(c3ccc(O)cc3)c3cc(O)ccc32)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GALR3 O60755 8/20 0.48
HTR4 Q13639 1/20 0.48
ESR1 P03372 6/20 0.43
ESR2 Q92731 4/20 0.43
ANPEP P15144 1/20 0.39
DPP4 P27487 1/20 0.39
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
THRB P10828 1/20 0.38
PKM P14618 1/20 0.38
BLM P54132 1/20 0.38
PLEC Q15149 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
APAF1 O14727 1/20 0.38
POLB P06746 1/20 0.38
BRD4 O60885 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12852971 0.91 GALR3 (0.60) GALR3HTR4MAPT
SCHEMBL8273687 0.85 GALR3 (0.69) GALR3HTR4
SCHEMBL8451954 0.83 GALR3 (0.46) GALR3HTR4ESR1ESR2APAF1
SCHEMBL917357 0.80 GALR3 (0.72) GALR3HTR4MAPT
SCHEMBL917358 0.80 GALR3 (0.72) GALR3HTR4MAPT
SCHEMBL5356363 0.80 GALR3 (0.78) GALR3HTR4
SCHEMBL5356357 0.80 GALR3 (0.78) GALR3HTR4
SCHEMBL8251705 0.80 GALR3 (0.46) GALR3HTR4ESR1ESR2APAF1
SCHEMBL8244088 0.79 GALR3 (0.49) GALR3HTR4MAPT
SCHEMBL8250355 0.77 TTR (0.61) GALR3HTR4KDM4EMAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7166635-B2 3-imino-2-indolones for the treatment of depression and/or anxiety H. LUNDBECK A/S (DK) 2007-01-23 US disclosed
US-20050148635-A1 3-imino-2-indolones for the treatment of depression and/or anxiety SYNAPTIC PHARMACEUTICAL CORPORATION 2005-07-07 US disclosed
US-20040082615-A1 3-Imino-2-indolones for the treatement of depression and/or anxiety H. LUNDBECK A/S (DK) 2004-04-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050148635-A1 3-imino-2-indolones for the treatment of depression and/or anxiety GALR3, GALR2, GALR1 GALR3 1/4885HTR4 17/4885ESR1 1020/4885
US-20040082615-A1 3-Imino-2-indolones for the treatement of depression and/or anxiety GALR3, GALR2, GALR1 GALR3 1/4885HTR4 13/4885ESR1 914/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.