SCHEMBL8250435

SCHEMBL8250435

CCOC(=O)C(Cc1ccc(NC(=O)c2c(Cl)cncc2Cl)cc1)NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 16/20 0.59
ITGB1 P05556 10/20 0.59
CYP3A4 P08684 1/20 0.54
NPC1 O15118 1/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13913379 0.87 CYP3A4 (0.64) ITGA4ITGB1CYP3A4
SCHEMBL4316900 0.87 CYP3A4 (0.64) ITGA4ITGB1CYP3A4
SCHEMBL13932617 0.87 CYP3A4 (0.51) ITGA4ITGB1CYP3A4
SCHEMBL13913382 0.86 ITGA4 (0.48) ITGA4ITGB1CYP3A4
SCHEMBL8259983 0.86 ITGA4 (0.48) ITGA4ITGB1CYP3A4
SCHEMBL6743406 0.85 ITGB1 (0.50) ITGA4ITGB1NPC1MEN1KMT2A
SCHEMBL750225 0.84 KMT2A (0.53) NPC1MEN1KMT2A
SCHEMBL13913390 0.83 ITGA4 (0.57) ITGA4ITGB1CYP3A4
SCHEMBL4316611 0.82 ITGB1 (0.59) ITGA4ITGB1
SCHEMBL13913372 0.82 ITGB1 (0.59) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006113199-A1 VLA-4 ANTAGONISTS MERCK & CO., INC. (US) 2006-10-26 WO disclosed