SCHEMBL8250765

SCHEMBL8250765

C[C@H](CO)NC(=O)CN1CCC(F)(CNC(=O)c2cc(O)cc(Cl)c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 14/20 0.56
CACNA1I Q9P0X4 5/20 0.47
SCN5A Q14524 1/20 0.47
CACNA1H O95180 4/20 0.39
CYP2D6 P10635 2/20 0.39
CACNA1G O43497 1/20 0.38
SMYD3 Q9H7B4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2886970 0.79 KCNH2 (0.88) KCNH2CACNA1ISCN5ACACNA1HCYP2D6
SCHEMBL5067690 0.78 KCNH2 (0.51) KCNH2CACNA1ISCN5ACACNA1HCACNA1G
SCHEMBL2888815 0.77 KCNH2 (0.73) KCNH2CACNA1ISCN5ACACNA1HCYP2D6
SCHEMBL2881952 0.76 KCNH2 (0.69) KCNH2CACNA1ISCN5ACACNA1HCYP2D6
SCHEMBL2889178 0.75 KCNH2 (0.73) KCNH2CACNA1ISCN5ACACNA1HCYP2D6
SCHEMBL8250567 0.75 KCNH2 (0.53) KCNH2CACNA1ISCN5ACACNA1HCYP2D6
SCHEMBL8243948 0.75 KCNH2 (0.63) KCNH2CACNA1ISCN5ACACNA1HCYP2D6
SCHEMBL2885430 0.74 KCNH2 (0.72) KCNH2CACNA1ISCN5ACACNA1HCYP2D6
SCHEMBL2889949 0.74 KCNH2 (0.72) KCNH2CACNA1ISCN5ACACNA1HCYP2D6
SCHEMBL2887799 0.74 KCNH2 (0.79) KCNH2CACNA1ISCN5ACACNA1HCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007002884-A2 4-FLUORO-PIPERIDINE T-TYPE CALCIUM CHANNEL ANTAGONISTS MERCK & CO., INC. (US) 2007-01-04 WO disclosed