SCHEMBL8251395

SCHEMBL8251395

COc1ccc2[nH]cc(CC(NC(=O)OC(C)(C)C)C(=O)N3CSCC3C(N)=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.45
TACR1 P25103 2/20 0.44
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
ACE P12821 1/20 0.42
CCKBR P32239 2/20 0.42
CTSL P07711 2/20 0.42
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HTR1A P08908 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
MMP2 P08253 1/20 0.41
MMP13 P45452 1/20 0.41
MMP14 P50281 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13814414 0.91 TACR1 (0.45) SCN9ATACR1HDAC1HDAC8ACE
SCHEMBL8243903 0.87 CTSL (0.47) SCN9ATACR1HDAC1HDAC8ACE
SCHEMBL4174694 0.84 CTSL (0.41) SCN9ATACR1HDAC1HDAC8ACE
SCHEMBL8939524 0.81 SCN9A (0.65) SCN9ATACR1ACECTSLCTSS
SCHEMBL8939526 0.81 SCN9A (0.65) SCN9ATACR1ACECTSLCTSS
SCHEMBL31407794 0.81 SCN9A (0.65) SCN9ATACR1ACECTSLCTSS
SCHEMBL4267961 0.79 SCN9A (0.46) SCN9ACCKBRMEN1KMT2A
SCHEMBL4108691 0.79 SCN9A (0.46) SCN9ACCKBRMEN1KMT2A
SCHEMBL31725820 0.79 TACR1 (0.61) SCN9ATACR1ACECTSLCTSS
SCHEMBL4265005 0.78 SCN9A (0.45) SCN9ACCKBRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006134613-A2 NOVEL 5-SUBSTITUTED INDOLE DERIVATIVES AS DIPEPTIDYL PEPTIDASE IV (DPP-IV) INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2006-12-21 WO disclosed