SCHEMBL8252265

SCHEMBL8252265

O=C(Nc1cccc(O)c1)Nc1cccc(C(=O)c2c[nH]c3ncccc23)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 2/20 0.51
CDC7 O00311 1/20 0.47
BRAF P15056 2/20 0.47
MAP2K1 Q02750 1/20 0.46
CLK1 P49759 1/20 0.45
DYRK1A Q13627 1/20 0.45
DYRK2 Q92630 1/20 0.45
DYRK1B Q9Y463 1/20 0.45
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.44
JAK3 P52333 1/20 0.44
RIPK1 Q13546 2/20 0.43
ROCK2 O75116 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
NPC1 O15118 1/20 0.42
STAT3 P40763 1/20 0.42
STAT1 P42224 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL411058 0.91 NEK2 (0.53) NEK2BRAFMAP2K1ALDH1A1HTT
SCHEMBL410517 0.89 ALDH1A1 (0.59) NEK2BRAFMAP2K1ALDH1A1HTT
SCHEMBL415660 0.89 NEK2 (0.51) NEK2BRAFMAP2K1ALDH1A1HTT
SCHEMBL857000 0.88 NEK2 (0.58) NEK2CDC7MAP2K1KMT2ARAB9A
SCHEMBL413384 0.88 TAAR1 (0.53) NEK2CDC7BRAFMAP2K1ALDH1A1
SCHEMBL416184 0.88 NPC1 (0.52) NEK2BRAFMAP2K1ALDH1A1HTT
SCHEMBL415961 0.88 BRAF (0.53) NEK2BRAFMAP2K1ALDH1A1HTT
SCHEMBL8247093 0.87 BRAF (0.52) NEK2BRAFRIPK1MEN1KMT2A
SCHEMBL414293 0.87 BRAF (0.55) NEK2BRAFMAP2K1CLK1DYRK1A
SCHEMBL410657 0.87 BRAF (0.62) NEK2BRAFMAP2K1ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007002325-A1 PYRROLO[2,3-B] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS PLEXXIKON, INC. (US) 2007-01-04 WO disclosed
WO-2007002433-A1 PYRROLO [2, 3-B] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS PLEXXIKON, INC. (US) 2007-01-04 WO disclosed