Aripiprazole

Aripiprazole

SCHEMBL8255

O=C1CCc2ccc(OCCCCN3CCN(c4cccc(Cl)c4Cl)CC3)cc2N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2HTR1AHTR2A

The experimentally established mechanism targets of Aripiprazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 20/20 1.00
HTR1A known ✓ P08908 3/20 1.00
HTR2A known ✓ P28223 3/20 1.00
DRD3 P35462 5/20 1.00
DRD4 P21917 4/20 1.00
HTR2B P41595 3/20 1.00
DRD1 P21728 2/20 1.00
DRD5 P21918 2/20 1.00
HTR2C P28335 2/20 1.00
HTR7 P34969 2/20 1.00
HTR6 P50406 2/20 1.00
HTR3E A5X5Y0 1/20 1.00
MEN1 O00255 1/20 1.00
MLNR O43193 1/20 1.00
HTR3B O95264 1/20 1.00
ABCB11 O95342 1/20 1.00
ESR1 P03372 1/20 1.00
PGR P06401 1/20 1.00
ADRB2 P07550 1/20 1.00
CHRM2 P08172 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Aripiprazole SCHEMBL29356997 1.00 DRD2 (1.00) DRD2DRD3DRD4HTR1AHTR2A
Aripiprazole SCHEMBL29475637 1.00 DRD2 (1.00) DRD2DRD3DRD4HTR1AHTR2A
Aripiprazole SCHEMBL29475638 1.00 DRD2 (1.00) DRD2DRD3DRD4HTR1AHTR2A
Aripiprazole SCHEMBL982189 1.00 DRD2 (1.00) DRD2DRD3DRD4HTR1AHTR2A
Aripiprazole SCHEMBL29438823 1.00 DRD2 (1.00) DRD2DRD3DRD4HTR1AHTR2A
Aripiprazole SCHEMBL7097505 0.99 DRD2 (0.98) DRD2DRD3DRD4HTR1AHTR2A
Aripiprazole SCHEMBL236666 0.99 DRD2 (0.98) DRD2DRD3DRD4HTR1AHTR2A
Aripiprazole SCHEMBL5147095 0.99 DRD2 (0.98) DRD2DRD3DRD4HTR1AHTR2A
Aripiprazole SCHEMBL30958766 0.99 DRD2 (0.98) DRD2DRD3DRD4HTR1AHTR2A
Aripiprazole SCHEMBL31174198 0.99 DRD2 (0.98) DRD2DRD3DRD4HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 30065 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260146048-A1 NOVEL BISINDOLYLMALEIMIDE KINASE INHIBITORS 4M THERAPEUTICS INC. (US) 2026-05-28 US claimed
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
CN-110204488-B Preparation method of lunar Gui Xiana risperidone SICHUAN KELUN PHARMACEUTICAL RESEARCH INSTITUTE Co.,Ltd. (CN) 2026-05-26 CN claimed
CN-122094963-A Cardioprotective lipids and methods of use 2026-05-26 CN claimed
CN-116199626-B Method for removing aripiprazole BQB impurities ZHEJIANG HUAHAI PHARMACEUTICAL CO.,LTD. (CN) 2026-05-26 CN claimed
CN-122079853-A N-substituted indoles and other heterocyclic compounds for the treatment of brain diseases 2026-05-26 CN claimed
WO-2026102521-A1 USE OF A PURINE COMPOUND FOR THE TREATMENT OF AUTISM SPECTRUM DISORDER, RETT SYNDROME, AND FRAGILE X SYNDROME MARVEL BIOTECHNOLOGY (CA) 2026-05-21 WO claimed
US-12629366-B2 Pharmaceutical compositions comprising sorbitan esters ALKERMES PHARMA IRELAND LIMITED (IE) 2026-05-19 US claimed
EP-4740962-A1 PHARMACEUTICAL COMPOSITION, FORMULATION CONTAINING PHARMACEUTICAL COMPOSITION, KIT CONTAINING PHARMACEUTICAL COMPOSITION, PREPARATION METHOD FOR PHARMACEUTICAL COMPOSITION, AND USE OF PHARMACEUTICAL COMPOSITION Shanghai WD Pharmaceutical Co., Ltd (CN) 2026-05-13 EP claimed
US-12624036-B2 Method of treating post-traumatic stress disorder INTRA-CELLULAR THERAPIES, INC. (US) 2026-05-12 US claimed
US-20020076437-A1 Flashmelt oral dosage formulation BRISTOL-MYERS SQUIBB COMPANY 2002-06-20 US claimed
WO-2002033112-A2 PROTEIN-PROTEIN INTERACTIONS IN NEURODEGENERATIVE DISEASES MYRIAD GENETICS, INC. (US) 2002-04-25 WO claimed
EP-1145711-A1 Flash-melt oral dosage formulation BRISTOL-MYERS SQUIBB COMPANY (US) 2001-10-17 EP claimed
CN-1317309-A Instant oral medincinal preparation BRISTOL MYERS SQUIBB CO (US) 2001-10-17 CN claimed
EP-0782692-A1 SENSOR ARRANGEMENT AND METHOD OF DETECTING MEASURED VALUES USING SAID SENSOR ARRANGEMENT Micro-Epsilon Messtechnik GmbH & Co. KG (DE) 1997-07-09 EP claimed
WO-1996009516-A1 SENSOR ARRANGEMENT AND METHOD OF DETECTING MEASURED VALUES USING SAID SENSOR ARRANGEMENT MICRO-EPSILON MESSTECHNIK GMBH & CO. KG (DE) 1996-03-28 WO claimed
EP-0367141-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1996-01-10 EP claimed
US-5006528-A Carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-04-09 US claimed
EP-0367141-A2 Carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-05-09 EP claimed
EP-0228345-A1 Magnetic-release mechanism for an earth fault circuit breaker CMC Carl Maier + Cie AG (CH) 1987-07-08 EP claimed