SCHEMBL8256099

SCHEMBL8256099

CC(=O)COCCOCCNC(=O)COCCOCCNC(=O)CC[C@@H](NC(=O)C(C)(C)CC(C)(C)C(=O)O)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GLP1R P43220 8/20 0.47
FOLH1 Q04609 7/20 0.31
CCKAR P32238 1/20 0.30
CCKBR P32239 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25862215 0.90 GLP1R (0.59) GLP1RCCKARCCKBR
SCHEMBL25462505 0.89 GLP1R (0.45) GLP1RFOLH1
SCHEMBL27342282 0.89 GLP1R (0.45) GLP1RFOLH1
SCHEMBL27343320 0.89 GLP1R (0.61) GLP1RFOLH1
SCHEMBL27343704 0.84 GLP1R (0.51) GLP1RFOLH1CCKARCCKBR
SCHEMBL71109 0.82 GLP1R (0.57) GLP1RFOLH1CCKARCCKBR
SCHEMBL20993544 0.82 GLP1R (0.50) GLP1RFOLH1
SCHEMBL72060 0.82 GLP1R (0.57) GLP1RFOLH1CCKARCCKBR
SCHEMBL71091 0.82 GLP1R (0.57) GLP1RFOLH1CCKARCCKBR
SCHEMBL24920301 0.81 GLP1R (0.45) GLP1RFOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2322546-A1 Acylated GLP-1 compounds NOVO NORDISK A/S (DK) 2011-05-18 EP disclosed
WO-2006097537-A2 ACYLATED GLP-1 COMPOUNDS NOVO NORDISK A/S (DK) 2006-09-21 WO disclosed
WO-2006097538-A1 EXTENDED GLP-1 COMPOUNDS NOVO NORDISK A/S (DK) 2006-09-21 WO disclosed