SCHEMBL8258555

SCHEMBL8258555

COCCCN1CCOc2ccc(CO[C@H]3CNC(CC(C)(C)C(=O)N(C)C)CC3c3ccc(OC)cc3)cc21

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
REN P00797 4/20 0.34
RORC P51449 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
THRB P10828 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2925854 1.00 REN (0.34) RENRORCALDH1A1CYP3A4CYP2D6
SCHEMBL2922315 0.95 REN (0.37) RENRORC
SCHEMBL2924373 0.93 REN (0.32) REN
SCHEMBL3550462 0.93 REN (0.34) RENRORCALDH1A1CYP3A4CYP2D6
SCHEMBL8258484 0.93 REN (0.34) RENRORCALDH1A1CYP3A4CYP2D6
SCHEMBL2947415 0.93 REN (0.34) RENRORCALDH1A1CYP3A4CYP2D6
SCHEMBL2923670 0.91 REN (0.34) RENRORCALDH1A1CYP3A4CYP2D6
SCHEMBL8473762 0.91 REN (0.34) RENRORCALDH1A1CYP3A4CYP2D6
SCHEMBL2922006 0.91 REN (0.34) RENRORCALDH1A1CYP3A4CYP2D6
SCHEMBL8257866 0.91 REN (0.35) RENRORCALDH1A1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1958634-A2 Substituted piperidines as inhibitors of beta-secretase, cathepsin D, plasmepsin II and/or HIV protease Speedel Experimenta AG (CH) 2008-08-20 EP disclosed
WO-2006103277-A2 2 , 4 , 5-SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS SPEEDEL EXPERIMENTA AG (CH) 2006-10-05 WO disclosed