SCHEMBL8259003

SCHEMBL8259003

O=C(CCCc1ccccc1)N[C@@H](Cc1ccccc1)C(=O)Nc1ccc2sc(C(=O)NO)cc2c1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 14/20 0.60
HDAC8 Q9BY41 2/20 0.51
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
HDAC9 Q9UKV0 1/20 0.49
HDAC5 Q9UQL6 1/20 0.49
CALCRL Q16602 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8260770 0.94 HDAC1 (0.63) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL5805384 0.90 HDAC1 (0.61) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL8255855 0.90 HDAC1 (0.61) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL8260757 0.88 HDAC1 (0.57) HDAC1
SCHEMBL5806429 0.88 HDAC1 (0.57) HDAC1
SCHEMBL8258701 0.87 HDAC1 (0.75) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL8259001 0.86 HDAC1 (0.67) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL5809231 0.86 HDAC1 (0.67) HDAC1HDAC8HDAC3HDAC4HDAC7
SCHEMBL5823705 0.86 HDAC1 (0.62) HDAC1
SCHEMBL8261102 0.86 HDAC1 (0.62) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006101454-A1 BENZOTHIOPHENE DERIVATIVES: PREPARATION AND PHARMACEUTICAL APPLICATIONS S*BIO PTE LTD (SG) 2006-09-28 WO disclosed