SCHEMBL8259643

SCHEMBL8259643

Cc1nnc(N2CC3=CC=CCC3C2)n1-c1ccc(Cl)cc1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 4/20 0.38
BRD4 O60885 11/20 0.37
OXTR P30559 4/20 0.35
TRPA1 O75762 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.33
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 1/20 0.32
BRD2 P25440 1/20 0.31
BRD3 Q15059 1/20 0.31
BRDT Q58F21 1/20 0.31
CREBBP Q92793 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8257678 0.83 AVPR1A (0.41) AVPR1AOXTR
SCHEMBL8258677 0.80 AVPR1A (0.31) AVPR1A
SCHEMBL8252339 0.76 AVPR1A (0.36) AVPR1ABRD4OXTR
SCHEMBL29163640 0.71 NOTUM (0.39) AVPR1AKMT2AKDM4E
SCHEMBL4620922 0.71 BRD4 (0.46) AVPR1ABRD4OXTRTRPA1TRPM8
SCHEMBL8256810 0.69 AVPR1A (0.48) AVPR1ABRD4OXTRTRPA1TRPM8
SCHEMBL5155966 0.69 AVPR1A (0.48) AVPR1ABRD4OXTRTRPA1TRPM8
SCHEMBL8285404 0.68 ADRB1 (0.56) AVPR1ABRD4TRPA1TRPM8
Hydrochloric Acid SCHEMBL315285 0.68 AVPR1A (0.47) AVPR1ABRD4OXTRTRPA1TRPM8
Hydrochloric Acid SCHEMBL5156223 0.68 AVPR1A (0.47) AVPR1ABRD4OXTRTRPA1TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006123242-A1 1, 2, 4 -TRIAZOLE DERIVATIVES AS VASOPRESSIN ANTAGONISTS PFIZER LIMITED (GB) 2006-11-23 WO disclosed