SCHEMBL825985

SCHEMBL825985

Nc1nc(OC2CCOC2)c2nc(-c3ccc(NC(=O)C4CCNC4)c(F)c3)ccc2n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.36
HDAC2 Q92769 5/20 0.36
MET P08581 2/20 0.36
ROCK2 O75116 1/20 0.35
JAK2 O60674 1/20 0.35
JAK3 P52333 1/20 0.35
GRM4 Q14833 2/20 0.34
HDAC3 O15379 2/20 0.34
RPS6KB1 P23443 1/20 0.34
MAPK8 P45983 1/20 0.34
MAPK9 P45984 1/20 0.34
PIK3CA P42336 2/20 0.33
MTOR P42345 2/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
PARP1 P09874 1/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
TTK P33981 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL823702 1.00 HDAC1 (0.36) HDAC1HDAC2METROCK2JAK2
SCHEMBL823651 0.88 JAK2 (0.45) HDAC1HDAC2JAK2JAK3GRM4
SCHEMBL825711 0.88 JAK2 (0.45) HDAC1HDAC2JAK2JAK3GRM4
SCHEMBL823650 0.85 PIK3CA (0.37) GRM4MAPK8MAPK9PIK3CAMTOR
SCHEMBL825938 0.85 PIK3CA (0.37) GRM4MAPK8MAPK9PIK3CAMTOR
SCHEMBL4423835 0.80 MAPK1 (0.46) JAK2GRM4MAPK8MAPK9PIK3CA
SCHEMBL4423840 0.80 ALOX5AP (0.38) HDAC1HDAC2GRM4MAPK8MAPK9
SCHEMBL3609814 0.76 HDAC1 (0.39) HDAC1HDAC2GRM4PIK3CAMTOR
SCHEMBL3605007 0.76 HDAC1 (0.39) HDAC1HDAC2GRM4PIK3CAMTOR
SCHEMBL13500401 0.76 HDAC1 (0.39) HDAC1HDAC2GRM4PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143394-B2 Pyrido(3,2-d)pyrimidines useful for treating viral infections GILEAD SCIENCES, INC. (US) 2012-03-27 US disclosed