SCHEMBL8260842

SCHEMBL8260842

CNC1(C)CCCc2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 3/20 0.53
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
AKR1B1 P15121 1/20 0.41
SIGMAR1 Q99720 2/20 0.41
HDAC9 Q9UKV0 1/20 0.41
EBP Q15125 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18088803 0.89 KDM1A (0.44) KDM1AHDAC9
SCHEMBL13198414 0.89 KDM1A (0.44) KDM1AHDAC9
SCHEMBL19577941 0.80 KDM1A (0.47) KDM1AMEN1KMT2AAKR1B1SIGMAR1
SCHEMBL11750121 0.79 KDM1A (0.44) KDM1AMEN1KMT2AAKR1B1SIGMAR1
SCHEMBL18088622 0.78 KDM1A (0.46) KDM1AMEN1KMT2AAKR1B1
SCHEMBL21376364 0.78 KDM1A (0.46) KDM1AMEN1KMT2AAKR1B1SIGMAR1
SCHEMBL10483582 0.76 KDM1A (0.51) KDM1AMEN1KMT2AAKR1B1SIGMAR1
SCHEMBL29556050 0.76 KDM1A (0.59) KDM1AMEN1KMT2AAKR1B1SIGMAR1
SCHEMBL578812 0.76 KDM1A (0.59) KDM1AMEN1KMT2AAKR1B1SIGMAR1
SCHEMBL2590935 0.76 HTR2A (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006102308-A2 BETA-LACTAMYL VASOPRESSIN V1B ANTAGONISTS AZEVAN PHARMACEUTICALS, INC. (US) 2006-09-28 WO disclosed