SCHEMBL8260880

SCHEMBL8260880

COc1ccc(C(=O)CC(C)C)cc1OCCCOC(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.48
PDE4B Q07343 6/20 0.44
SMPD1 P17405 4/20 0.44
PRSS1 P07477 2/20 0.44
PDE4A P27815 1/20 0.43
PDE4C Q08493 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2438091 0.86 PDE4D (0.53) PDE4DPDE4BSMPD1PRSS1
SCHEMBL2439225 0.84 PDE4D (0.53) PDE4DPDE4BSMPD1
SCHEMBL3375161 0.84 CA12 (0.58) PDE4DPDE4BSMPD1PRSS1PDE4A
SCHEMBL29555877 0.80 PDE4D (0.62) PDE4DPDE4BPDE4APDE4C
SCHEMBL11045658 0.80 PDE4D (0.62) PDE4DPDE4BPDE4APDE4C
SCHEMBL2441538 0.75 PDE4D (0.57) PDE4DPDE4BPDE4APDE4C
SCHEMBL2592347 0.75 TSHR (0.62) PRSS1
SCHEMBL13433959 0.74 L3MBTL1 (0.52)
SCHEMBL2589912 0.74 MAPT (0.55) SMPD1PRSS1
SCHEMBL16930080 0.73 SMPD1 (0.51) PDE4DPDE4BSMPD1PRSS1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006100036-A1 3, 4-SUBSTITUTED PYRROLIDINE DERIVATIVES FOR THE TREATMENT OF HYPERTENSION NOVARTIS AG (CH) 2006-09-28 WO disclosed