SCHEMBL8273121

SCHEMBL8273121

COC(=O)c1cc(I)oc1CBr

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.36
ALDH1A1 P00352 7/20 0.36
KDM4E B2RXH2 6/20 0.36
HPGD P15428 3/20 0.36
HSD17B10 Q99714 3/20 0.35
CA12 O43570 3/20 0.35
CA2 P00918 3/20 0.35
CA7 P43166 3/20 0.35
CA9 Q16790 3/20 0.35
CA14 Q9ULX7 3/20 0.35
CA1 P00915 2/20 0.35
PDK2 Q15119 1/20 0.35
PDK4 Q16654 1/20 0.35
MAPT P10636 3/20 0.35
GAA P10253 2/20 0.35
TSHR P16473 2/20 0.35
ALOX15 P16050 1/20 0.35
CFTR P13569 1/20 0.35
CA3 P07451 1/20 0.35
CA6 P23280 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8273124 0.85 CA12 (0.41) ALDH1A1KDM4EHPGDHSD17B10CA12
SCHEMBL1674226 0.81 KMT2A (0.41) ALDH1A1KDM4EHPGDHSD17B10CA12
SCHEMBL2840089 0.78 MAPK1 (0.54) ALDH1A1KDM4EHSD17B10MAPTGAA
SCHEMBL8273120 0.75 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDHSD17B10CA12
SCHEMBL26985505 0.75 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDHSD17B10CA12
SCHEMBL8273126 0.71 ALDH1A1 (0.40) SOS1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL26985518 0.69 GAA (0.36) ALDH1A1KDM4EHPGDCA2CA9
SCHEMBL5860698 0.69 KDM4E (0.46) ALDH1A1KDM4EHSD17B10MAPTGAA
SCHEMBL2109561 0.69 HSD17B10 (0.44) ALDH1A1KDM4EHPGDHSD17B10CA12
SCHEMBL23577866 0.69 SOS1 (0.41) SOS1ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7511062-B2 Substituted 2-quinolyl-oxazoles useful as PDE4 inhibitors SCHERING CORPORATION (US) 2009-03-31 US disclosed
US-7511062-B2 Substituted 2-quinolyl-oxazoles useful as PDE4 inhibitors SCHERING CORPORATION (US) 2009-03-31 US disclosed
WO-2005116009-A1 SUBSTITUTED 2-QUINOLYL-OXAZOLES USEFUL AS PDE4 INHIBITORS SCHERING CORPORATION (US) 2005-12-08 WO disclosed