SCHEMBL8275502

SCHEMBL8275502

Cc1c(C(=O)NCCc2ccccc2)[nH]c2ccc([S+]([O-])N3CC(C)CC(C)C3)cc12

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.51
EGFR P00533 4/20 0.49
CDK2 P24941 4/20 0.49
CNR1 P21554 5/20 0.47
CNR2 P34972 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
LMNA P02545 1/20 0.46
RAB9A P51151 1/20 0.46
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CAPN1 P07384 1/20 0.41
MCL1 Q07820 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10259162 0.82 CNR1 (0.68) PTGS2EGFRCDK2CNR1CNR2
SCHEMBL8277185 0.81 PTGS2 (0.49) PTGS2EGFRCDK2CNR1CNR2
SCHEMBL8276724 0.77 CNR1 (0.61) PTGS2CNR1CNR2SMN1; SMN2LMNA
SCHEMBL10261543 0.75 HTT (0.55) PTGS2EGFRCDK2CNR1CNR2
SCHEMBL10262091 0.73 CNR1 (0.67) CNR1CNR2SMN1; SMN2LMNAMEN1
SCHEMBL10261074 0.70 BACE1 (0.55) PTGS2EGFRCDK2CNR1CNR2
SCHEMBL10261057 0.67 CNR1 (0.53) CNR1CNR2SMN1; SMN2LMNAMEN1
SCHEMBL20795007 0.67 PTGS2 (0.55) PTGS2EGFRCDK2CNR1CNR2
SCHEMBL20794349 0.66 PTGS2 (0.54) PTGS2EGFRCDK2CNR1CNR2
SCHEMBL10293115 0.66 CNR1 (0.60) CNR1CNR2NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006010008-A1 HETEROCYCLIC DERIVATIVES FOR MODULATION OF CALCIUM CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-26 WO disclosed